Tryptase g1 Protease Assay for compound screening and profiling via fluorescence-based quantification of enzyme activity.
Target Overview
CAT#
Tryptase g1
Enzyme
Human Tryptase gamma 1
Synonym
TPSG1, Serine protease 31, Transmembrane tryptase
Substrates
Fluorogenic substrate Mca-RPKPVE-Nval-WRK(Dnp)-NH2, 5 µM
Assay Properties
Readout
Enzymatic activity
Reference Compound IC50s
| Compounds | IC50 (µM) |
|---|---|
| Gabexate Mesylate | 3.9 |
| Leupeptin | 1.5 |
Scientific Information
Screening Location
Malvern, PA, USA
Further information
More information can be found on our website Protease Assay Services.
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