cGAS (AA 157-522) SPR Assay Service

Nucleotidyltransferase cGAS (AA 157-522) assay with surface plasmon resonance (SPR) technique

Target Overview

Target

Human cGAS fragment (AA 157-522)

HGNC symbol

CGAS (AA 157-522)

Synonyms

Cyclic GMP-AMP synthase, cGAMP synthase

Scientific information

Screening location

Malvern, PA, USA

Further information

More information can be found on our website SPR Assay Services for Drug Discovery

Binding kinetics and steady state affinity of PF-06928215 to cGAS (aa157-522)

cGAS SPR kinetics
cGAS SPR steady state

 

The data was collected on a Biacore 8K using multi-cycle kinetics. cGAS (AA 157-522) was immobilized to the sensor chip and the binding of PF-06928215 was measured. The binding data was analyzed using both a 1:1 kinetic binding model and a steady state affinity model.