BAZ1B-His Reader Domain Assay for compound screening and profiling using the AlphaScreen assay format to measure compound binding to the target.
Target Overview
CAT#
BAZ1B-His
Enzyme
Human BAZ1B-His
Synonyms
Bromodomain adjacent to zinc finger domain protein 1B, hWALp2, WBSC10, WBSCR10, WBSCR9, WSTF
Substrates
Histone H4 peptide (1-21) K5/8/12/16Ac
Assay Properties
Reaction
AlphaScreen Binding assay
Readout
Fluorescence
Reference Compound IC50s
| Compounds | IC50 (nM) |
|---|---|
| JQ-1 | 21,000 |
| SGC-CBP30 | 23,000 |
| GSK2801 | 70,000 |
Scientific Information
Q9UIG0 (http://www.uniprot.org/uniprot/Q9UIG0)
Screening Location
Malvern, USA
Further information
More information can be found on our website Reader Domain Assay Services.
Reference Compound IC50 for BAZ1B
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