BAZ2B-His Reader Domain Assay for compound screening and profiling using the AlphaScreen assay format to measure compound binding to the target.
Target Overview
CAT#
BAZ2B-His
Enzyme
Human BAZ2B-His
Synonyms
Bromodomain adjacent to zinc finger domain protein 2B, hWALp4, KIAA1476
Substrates
Histone H3 peptide (1-21) K9/14Ac
Assay Properties
Reaction
AlphaScreen Binding assay
Readout
Fluorescence
Reference Compound IC50s
| Compounds | IC50 (nM) |
|---|---|
| JQ-1 | 84,000 |
| Bromosporine | 85,000 |
| SGC-CBP30 | 105,000 |
| GSK2801 | 534 |
Scientific Information
Scientific Information: Q9UIF8 (http://www.uniprot.org/uniprot/Q9UIF8)
Screening Location
Malvern, USA
Further information
More information can be found on our website Reader Domain Assay Services.
Reference Compound IC50 for BAZ2B
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