Furin Protease Assay for compound screening and profiling via fluorescence-based quantification of enzyme activity.
Target Overview
CAT#
Furin
Enzyme
Human Furin
Synonym
FUR, PACE, PCSK3
Substrates
Fluorogenic peptide [pERTKR -AMC], 5 μM
Assay Properties
Readout
Enzymatic activity
Reference Compound IC50s
| Compounds | IC50 (nM) |
|---|---|
| Furin Inhibitor 1 | 1.6 |
| Furin Inhibitor 2 | 110 |
Scientific Information
P09958 (http://www.uniprot.org/uniprot/P09958)
Screening Location
Malvern, USA
Further information
More information can be found on our website Protease Assay Services.
Reference compound IC50 for Furin
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